Search Ontology:
ChEBI

dabrafenib mesylate

Term ID
CHEBI:75048
Synonyms
  • dabrafenib monomesylate
  • GSK 2118436
  • GSK 2118436B
  • N-{3-[5-(2-aminopyrimidin-4-yl)-2-tert-butyl-1,3-thiazol-4-yl]-2-fluorophenyl}-2,6-difluorobenzenesulfonamide methanesulfonate
  • Tafinlar
Definition
A methanesulfonate (mesylate) salt prepared from equimolar amounts of dabrafenib and methanesulfonic acid. Used for treatment of metastatic melanoma.
References
  • cas:1195768-06-9
  • kegg.drug:D10104
  • patent:WO2011047238
  • pubmed:23035153
  • pubmed:23102194
  • pubmed:23881668
  • reaxys:19690182
  • wikipedia.en:Dabrafenib
Ontology
ChEBI  ( EBI )
Relationships
Phenotype
Phenotype resulting from dabrafenib mesylate
Phenotype where environments contain dabrafenib mesylate
Phenotype modified by environments containing dabrafenib mesylate
Phenotype affecting dabrafenib mesylate
Human Disease Model