labetalol

Term ID

CHEBI:6343

Synonyms

• 2-hydroxy-5-{1-hydroxy-2-[(1-methyl-3-phenylpropyl)amino]ethyl}benzamide
• 3-Carboxamido-4-hydroxy-alpha-((1-methyl-3-phenylpropylamino)methyl)benzyl alcohol
• 5-(1-Hydroxy-2-(1-methyl-3-phenylpropylamino)ethyl)salicylamide
• kabetalol
• Labetalol
• labetalolum

Definition

A diastereoisomeric mixture of approximately equal amounts of all four possible stereoisomers ((R,S)-labetolol, (S,R)-labetolol, (S,S)-labetalol and (R,R)-labetalol). It is an adrenergic antagonist used to treat high blood pressure.

References

• Beilstein:2948416
• CAS:36894-69-6
• DrugBank:DB00598
• Drug_Central:1531
• HMDB:HMDB0014736
• KEGG:C07063
• KEGG:D08106
• LINCS:LSM-1282
• PMID:1447344
• PMID:16795017
• PMID:21908132
• PMID:22300487
• PMID:22528277
• PMID:23055089
• PMID:28166217
• PMID:31643185
• PMID:32709242
• PMID:33210850
• PMID:33424327
• PMID:33638710
• PMID:33893609
• PMID:34217067
• PMID:35075411
• PMID:7295463
• Patent:DE2032642
• Patent:US4012444
• Reaxys:2948416
• Wikipedia:Labetalol

Ontology

ChEBI  ( EBI )

Resources

CTD