Search Ontology:
ChEBI
pelabresib
- Term ID
- CHEBI:189653
- Synonyms
-
- 2-((4S)-6-(4-chlorophenyl)-1-methyl-4H-isoxazolo[5,4-d][2]benzazepin-4-yl)acetamide
- 2-[(4S)-6-(4-chlorophenyl)-1-methyl-4H-[1,2]oxazolo[5,4-d][2]benzazepin-4-yl]acetamide
- CPI 0610
- CPI-0610
- CPI-0610 anhydrous
- CPI-232
- CPI0610
- pelabresib
- pelabresibum
- Definition
- An organic heterotricyclic compound that is 4H-[1,2]oxazolo[5,4-d][2]benzazepine substituted by methyl, 2-amino-2-oxoethyl, and 4-chlorophenyl groups at positions 1, 4S and 6, respectively. It is a small molecule inhibitor of bromodomain and extra-terminal (BET) proteins and exhibits antineoplastic activity.
- References
-
- cas:1380087-89-7
- chemspider:32738784
- pubmed:26815195
- pubmed:27890933
- pubmed:30529073
- pubmed:31729905
- pubmed:32245330
- pubmed:32927276
- pubmed:33509905
- pubmed:33574760
- pubmed:33925695
- pubmed:35114569
- wikipedia.en:CPI-0610
- Ontology
- ChEBI ( EBI )
Phenotype
Phenotype resulting from pelabresib
Phenotype where environments contain pelabresib
Phenotype modified by environments containing pelabresib
Phenotype affecting pelabresib
Human Disease Model