Term Name: H1-receptor antagonist
Synonyms: classical antihistamines, classical antihistaminics, H1 antihistaminics, H1 receptor antagonists, H1 receptor blockaders, H1-receptor antagonists, H1-receptor blocker, H1-receptor blockers
Definition: H1-receptor antagonists are the drugs that selectively bind to but do not activate histamine H1 receptors, thereby blocking the actions of endogenous histamine.
Ontology: ChEBI [CHEBI:37955]  ( EBI )

Relationships
is a type of: histamine antagonist
inverse has_role: (S)-carbinoxamine maleate acrivastine alcaftadine antazoline aripiprazole aripiprazole lauroxil astemizole azatadine azatadine maleate azelastine azelastine hydrochloride benzquinamide benzylpenicillin clemizole bepotastine bepotastine besylate bromazine bromazine hydrochloride brompheniramine carbinoxamine carbinoxamine maleate cetirizine chlorphenamine cinnarizine clemastine clemastine fumarate clopenthixol cyclizine cyclizine hydrochloride cyproheptadine cyproheptadine hydrochloride sesquihydrate deptropine deptropine citrate desipramine desloratadine dexbrompheniramine dexbrompheniramine maleate dimenhydrinate diphenhydramine diphenhydramine hydrochloride diphenhydramine salicylate diphenylpyraline diphenylpyraline hydrochloride dithiadene doxylamine emedastine emedastine difumarate epinastine fexofenadine hydroxyzine ketotifen ketotifen fumarate loratadine mepyramine methapyrilene methapyrilene hydrochloride mianserin mirtazapine N-demethylmirtazapine orphenadrine orphenadrine citrate orphenadrine hydrochloride oxatomide paliperidone paliperidone palmitate pimozide promazine promethazine promethazine hydrochloride risperidone sertindole thioridazine trazodone trazodone hydrochloride triprolidine triprolidine hydrochloride (anh.) triprolidine hydrochloride monohydrate triprolidine(1+) zuclopenthixol