Term Name: AZ505
Synonyms: AZ 505, AZ-505, N-cyclohexyl-3-[2-(3,4-dichlorophenyl)ethylamino]-N-[2-[2-(5-hydroxy-3-oxo-4H-1,4-benzoxazin-8-yl)ethylamino]ethyl]propanamide, N-cyclohexyl-N(3)-[2-(3,4-dichlorophenyl)ethyl]-N-(2-{[2-(5-hydroxy-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-8-yl)ethyl]amino}ethyl)-beta-alaninamide
Definition: A benzoxazine that is 2H-1,4-benzoxazin-3(4H)-one substituted by a hydroxy group at position 5 and a 2-{[2-(cyclohexyl{N-[2-(3,4-dichlorophenyl)ethyl]-beta-alanyl}amino)ethyl]amino}ethyl group at position 8. It is a potent and selective inhibitor of SMYD2.
Ontology: ChEBI [CHEBI:228259]  ( EBI )

Relationships
is a type of: benzoxazine dichlorobenzene organic hydroxy compound secondary amino compound tertiary carboxamide
has_role: antineoplastic agent EC 2.1.1.354 ([histone H3]-lysine(4) N-trimethyltransferase) inhibitor